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2-Benzamido-N-(1H-benzo[d]imidazol-2-yl)thiazole-4-carboxamide derivatives as potent inhibitors of CK1 delta/epsilon

Erstveröffentlichung
2012
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Wissenschaftlicher Artikel


Authors
Bischof, Joachim
Leban, Johann
Zaja, Mirko
Grothey, Arnhild
Radunsky, Barbara
et al.
Institutions
UKU. Klinik für Allgemein- und Viszeralchirurgie
Published in
Amino Acids ; 43 (2012), 4. - S. 1577-1591. - ISSN 0939-4451. - eISSN 1438-2199
Link to publication
https://dx.doi.org/10.1007/s00726-012-1234-x
Keywords
CK1 delta; CK1 epsilon; Phosphorylation; Small molecule inhibitor; Crystal structure; MTT; FACS; NF-KAPPA-B; CARCINOMA CELL-LINE; KINASE-I FAMILY; RHEUMATOID-ARTHRITIS; PROTEIN; SITE; VIVO; P53; CASEIN-KINASE-1-DELTA
Dewey Decimal Group
DDC 570 / Life sciences

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